TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University of New Orleans
Curated by ChEMBL
University of New Orleans
Curated by ChEMBL
Affinity DataKi: 0.0500nMAssay Description:Displacement of [3H]citalopram from serotonin transporter in Sprague-Dawley rat brain after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University of New Orleans
Curated by ChEMBL
University of New Orleans
Curated by ChEMBL
Affinity DataKi: 0.0610nMAssay Description:Displacement of [3H]citalopram from SERT in rat brainMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
University of New Orleans
Curated by ChEMBL
University of New Orleans
Curated by ChEMBL
Affinity DataKi: 0.0790nMAssay Description:In vitro binding affinity by inhibiting [3H]cytisine binding in rat brain tissue at Nicotinic acetylcholine receptor alpha4-beta2More data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University of New Orleans
Curated by ChEMBL
University of New Orleans
Curated by ChEMBL
Affinity DataKi: 0.100nMAssay Description:Displacement of [3H]citalopram from SERT in rat brainMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
University of New Orleans
Curated by ChEMBL
University of New Orleans
Curated by ChEMBL
Affinity DataKi: 0.140nMAssay Description:in vitro binding affinity by inhibiting [3H]cytisine binding in rat brain tissue at Nicotinic acetylcholine receptor alpha4-beta2More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
University of New Orleans
Curated by ChEMBL
University of New Orleans
Curated by ChEMBL
Affinity DataKi: 0.160nMAssay Description:in vitro binding affinity by inhibiting [3H]cytisine binding in rat brain tissue at Nicotinic acetylcholine receptor alpha4-beta2More data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University of New Orleans
Curated by ChEMBL
University of New Orleans
Curated by ChEMBL
Affinity DataKi: 0.300nMAssay Description:Displacement of [3H]citalopram from SERT in rat brainMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University of New Orleans
Curated by ChEMBL
University of New Orleans
Curated by ChEMBL
Affinity DataKi: 0.600nMAssay Description:Displacement of [3H]citalopram from serotonin transporter in Sprague-Dawley rat brain after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University of New Orleans
Curated by ChEMBL
University of New Orleans
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Displacement of [3H]citalopram from serotonin transporter in Sprague-Dawley rat brain after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University of New Orleans
Curated by ChEMBL
University of New Orleans
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Displacement of [3H]Citalopram from SERT in Sprague-Dawley rat brain homogenate after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University of New Orleans
Curated by ChEMBL
University of New Orleans
Curated by ChEMBL
Affinity DataKi: 1.30nMAssay Description:Displacement of [3H]Citalopram from SERT in Sprague-Dawley rat brain homogenate after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University of New Orleans
Curated by ChEMBL
University of New Orleans
Curated by ChEMBL
Affinity DataKi: 1.70nMAssay Description:Displacement of [3H]citalopram from serotonin transporter in Sprague-Dawley rat brain after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University of New Orleans
Curated by ChEMBL
University of New Orleans
Curated by ChEMBL
Affinity DataKi: 1.80nMAssay Description:Displacement of [3H]citalopram from SERT in rat brainMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University of New Orleans
Curated by ChEMBL
University of New Orleans
Curated by ChEMBL
Affinity DataKi: 2nMAssay Description:Displacement of [3H]citalopram from serotonin transporter in Sprague-Dawley rat brain after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University of New Orleans
Curated by ChEMBL
University of New Orleans
Curated by ChEMBL
Affinity DataKi: 2nMAssay Description:Displacement of [3H]citalopram from serotonin transporter in Sprague-Dawley rat brain after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University of New Orleans
Curated by ChEMBL
University of New Orleans
Curated by ChEMBL
Affinity DataKi: 2nMAssay Description:Displacement of [3H]citalopram from serotonin transporter in Sprague-Dawley rat brain after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University of New Orleans
Curated by ChEMBL
University of New Orleans
Curated by ChEMBL
Affinity DataKi: 2.5nMAssay Description:Displacement of [3H]citalopram from serotonin transporter in Sprague-Dawley rat brain after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University of New Orleans
Curated by ChEMBL
University of New Orleans
Curated by ChEMBL
Affinity DataKi: 2.80nMAssay Description:Displacement of [3H]citalopram from SERT in rat brainMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University of New Orleans
Curated by ChEMBL
University of New Orleans
Curated by ChEMBL
Affinity DataKi: 2.90nMAssay Description:Displacement of [3H]Citalopram from SERT in Sprague-Dawley rat brain homogenate after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University of New Orleans
Curated by ChEMBL
University of New Orleans
Curated by ChEMBL
Affinity DataKi: 2.90nMAssay Description:Displacement of [3H]citalopram from serotonin transporter in Sprague-Dawley rat brain after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University of New Orleans
Curated by ChEMBL
University of New Orleans
Curated by ChEMBL
Affinity DataKi: 3nMAssay Description:Displacement of [3H]Citalopram from SERT in Sprague-Dawley rat brain homogenate after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University of New Orleans
Curated by ChEMBL
University of New Orleans
Curated by ChEMBL
Affinity DataKi: 3.30nMAssay Description:Displacement of [3H]citalopram from serotonin transporter in Sprague-Dawley rat brain after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University of New Orleans
Curated by ChEMBL
University of New Orleans
Curated by ChEMBL
Affinity DataKi: 3.5nMAssay Description:Displacement of [3H]Citalopram from SERT in Sprague-Dawley rat brain homogenate after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University of New Orleans
Curated by ChEMBL
University of New Orleans
Curated by ChEMBL
Affinity DataKi: 3.70nMAssay Description:Binding affinity at dopamine transporter from rat caudate-putamen tissue by [3H]-WIN- 35428 displacement.More data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University of New Orleans
Curated by ChEMBL
University of New Orleans
Curated by ChEMBL
Affinity DataKi: 3.90nMAssay Description:Displacement of [3H]citalopram from serotonin transporter in Sprague-Dawley rat brain after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University of New Orleans
Curated by ChEMBL
University of New Orleans
Curated by ChEMBL
Affinity DataKi: 3.90nMAssay Description:Displacement of [3H]WIN35428 from DAT in Sprague-Dawley rat brain homogenates after 1 hr by scintillation countingMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University of New Orleans
Curated by ChEMBL
University of New Orleans
Curated by ChEMBL
Affinity DataKi: 4nMAssay Description:Displacement of [3H]Citalopram from SERT in Sprague-Dawley rat brain homogenate after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University of New Orleans
Curated by ChEMBL
University of New Orleans
Curated by ChEMBL
Affinity DataKi: 4nMAssay Description:Displacement of [3H]WIN35428 from DAT in Sprague-Dawley rat brain homogenates after 1 hr by scintillation countingMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University of New Orleans
Curated by ChEMBL
University of New Orleans
Curated by ChEMBL
Affinity DataKi: 4.10nMAssay Description:Binding affinity at dopamine transporter from rat caudate-putamen tissue by [3H]-WIN- 35428 displacement.More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
University of New Orleans
Curated by ChEMBL
University of New Orleans
Curated by ChEMBL
Affinity DataKi: 4.20nMAssay Description:in vitro binding affinity by inhibiting [3H]cytisine binding in rat brain tissue at Nicotinic acetylcholine receptor alpha4-beta2More data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University of New Orleans
Curated by ChEMBL
University of New Orleans
Curated by ChEMBL
Affinity DataKi: 4.20nMAssay Description:Displacement of [3H]Citalopram from SERT in Sprague-Dawley rat brain homogenate after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University of New Orleans
Curated by ChEMBL
University of New Orleans
Curated by ChEMBL
Affinity DataKi: 4.30nMAssay Description:Displacement of [3H]citalopram from serotonin transporter in Sprague-Dawley rat brain after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 4.60nMAssay Description:Displacement of [3H]SR141716 from CB1 receptor in rat cerebellum homogenateMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University of New Orleans
Curated by ChEMBL
University of New Orleans
Curated by ChEMBL
Affinity DataKi: 4.70nMAssay Description:Displacement of [3H]citalopram from SERT in rat brainMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University of New Orleans
Curated by ChEMBL
University of New Orleans
Curated by ChEMBL
Affinity DataKi: 4.80nMAssay Description:Displacement of [3H]Citalopram from SERT in Sprague-Dawley rat brain homogenate after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University of New Orleans
Curated by ChEMBL
University of New Orleans
Curated by ChEMBL
Affinity DataKi: 4.90nMAssay Description:Displacement of [3H]WIN35428 from DAT in Sprague-Dawley rat brain homogenates after 1 hr by scintillation countingMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University of New Orleans
Curated by ChEMBL
University of New Orleans
Curated by ChEMBL
Affinity DataKi: 5.70nMAssay Description:Binding affinity at dopamine transporter from rat caudate-putamen tissue by [3H]-WIN- 35428 displacement.More data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University of New Orleans
Curated by ChEMBL
University of New Orleans
Curated by ChEMBL
Affinity DataKi: 5.90nMAssay Description:Displacement of [3H]citalopram from serotonin transporter in Sprague-Dawley rat brain after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University of New Orleans
Curated by ChEMBL
University of New Orleans
Curated by ChEMBL
Affinity DataKi: 5.90nMAssay Description:Displacement of [3H]citalopram from serotonin transporter in Sprague-Dawley rat brain after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University of New Orleans
Curated by ChEMBL
University of New Orleans
Curated by ChEMBL
Affinity DataKi: 6.10nMAssay Description:Displacement of [3H]citalopram from SERT in rat brainMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University of New Orleans
Curated by ChEMBL
University of New Orleans
Curated by ChEMBL
Affinity DataKi: 6.10nMAssay Description:Displacement of [3H]WIN35428 from DAT in Sprague-Dawley rat brain homogenates after 1 hr by scintillation countingMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University of New Orleans
Curated by ChEMBL
University of New Orleans
Curated by ChEMBL
Affinity DataKi: 6.40nMAssay Description:Displacement of [3H]citalopram from serotonin transporter in Sprague-Dawley rat brain after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University of New Orleans
Curated by ChEMBL
University of New Orleans
Curated by ChEMBL
Affinity DataKi: 7nMAssay Description:Displacement of [3H]citalopram from serotonin transporter in Sprague-Dawley rat brain after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University of New Orleans
Curated by ChEMBL
University of New Orleans
Curated by ChEMBL
Affinity DataKi: 7nMAssay Description:Displacement of [3H]WIN35428 from DAT in Sprague-Dawley rat brain homogenates after 1 hr by scintillation countingMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University of New Orleans
Curated by ChEMBL
University of New Orleans
Curated by ChEMBL
Affinity DataKi: 7.20nMAssay Description:Inhibition of [3H]paroxetine binding to rat serotonin transporterMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University of New Orleans
Curated by ChEMBL
University of New Orleans
Curated by ChEMBL
Affinity DataKi: 7.20nMAssay Description:Displacement of [3H]citalopram from serotonin transporter in Sprague-Dawley rat brain after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University of New Orleans
Curated by ChEMBL
University of New Orleans
Curated by ChEMBL
Affinity DataKi: 7.20nMAssay Description:Displacement of [3H]-paroxetine from serotonin transporter (SERT)More data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University of New Orleans
Curated by ChEMBL
University of New Orleans
Curated by ChEMBL
Affinity DataKi: 7.30nMAssay Description:Displacement of [3H]Citalopram from SERT in Sprague-Dawley rat brain homogenate after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University of New Orleans
Curated by ChEMBL
University of New Orleans
Curated by ChEMBL
Affinity DataKi: 7.40nMAssay Description:Binding affinity at dopamine transporter from rat caudate-putamen tissue by [3H]-WIN- 35428 displacement.More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University of New Orleans
Curated by ChEMBL
University of New Orleans
Curated by ChEMBL
Affinity DataKi: 7.60nMAssay Description:Displacement of [3H]WIN35428 from DAT in Sprague-Dawley rat brain homogenates after 1 hr by scintillation countingMore data for this Ligand-Target Pair